Content
For the treatment of hormonal disorders in men, testosterone preparations are used, which are presented in pharmacies in tablets and solutions. Medicines are hormonal. Testosterone plays an important role in the body, so its deficiency or excess significantly affects the quality of life. Over time, a man begins to feel deviations in the amount of this hormone from the norm, which is manifested by unpleasant symptoms. Pharmaceutical testosterone helps to correct the hormonal background.
What is testosterone
This is the name of one of the most important hormones of metabolism, which is part of many metabolic processes. For each period of human development, there is a base level of testosterone. The original form of this sex hormone is not very active due to binding to androgen receptors and a protein that transports the substance in the blood. It acquires a working appearance under the action of the enzyme 5-alpha-reductase. It is produced by the adrenal cortex and testicles. The synthesis is influenced by the follicle-stimulating and luteinizing hormone of the pituitary gland.
Leading testosterone is in the processes that relate to the reproductive system. It is necessary for the formation of secondary sexual characteristics, attraction, development of male gonads and spermatogenesis. Other properties:
- regulation of weight and mood;
- increase in muscle mass;
- the formation of memory and the ability to learn.
How to increase testosterone in men
There are a large number of medications that lead to an increase in the level of this hormone. In general, they can be divided into two groups depending on the mechanism of action:
- Pharmaceutical preparations for increasing testosterone in men using hormone replacement therapy. This method of treatment involves the elimination of the deficiency of the specified hormone by replacing exogenous synthetic or natural analogues. This method contributes to the rapid solution of the problem. The downside is the need to continue to use a synthetic hormone.
- Drugs that stimulate the natural production of testosterone. Medicines from this group are able to activate the work of their own endocrine glands. This method of treatment is longer, but more effective than the previous one. The body independently produces the right amount of such an important hormone for a man. Especially often this method is used in the treatment of young patients.
Male hormones in tablets
Compared to injectables, testosterone tablets are a more convenient type of drug treatment. This is especially true for those who are contraindicated injections. A feature of the application is the need to drink tablets every day. The therapeutic effect of such therapy develops faster. The drug increases potency and sexual function in general.
The disadvantage is that the active substance is not retained for a long time by the body. For this reason, the quickly onset effect also passes quickly. Popular drugs to increase testosterone in men in this category:
- Andriol;
- Halotestin;
- Proviron;
- Vistimon;
- Metadren.
Testosterone Stimulants
Preparations from this group activate the corresponding processes that force the body to independently produce the required amount of sex hormone. It is worth noting here that treatment with stimulants does not always bring the desired effect. The reason is the individual characteristics of the reserves of the body of each man. Stimulants are often used to build muscle mass or enhance male potency.
The principle of action involves the activation of the production of luteinizing enzyme. It affects the testicles, which, after receiving the signal, begin to produce the sex hormone. The following drugs have this effect:
- Arimatest;
- Vitrix;
- Cyclo-Bolan;
- Animal Test;
- Evo Test.
Even the fact that stimulants are not hormonal drugs does not negate prior consultation with a doctor before taking them. In order for their therapy to be truly effective, it is important to adhere to the instructions and dosage. Before the appointment of stimulants, it is necessary to conduct tests for hormones, because treatment with hormonal drugs may be required. Self-medication with stimulants can cause negative consequences.
Supplements to increase testosterone in men
Preparations of the category of dietary supplements are not drugs, like hormone replacements, but they are also able to increase the level of sex hormones. It is worth noting here that such supplements cannot treat serious hormonal disorders. Serious complications can result. For this reason, taking dietary supplements is recommended for those who want to build muscle mass and increase sexual arousal. Most often, these funds are used in bodybuilding by professional athletes.
You can not hope for a hundred percent result from taking dietary supplements. They are not tested in a clinical setting. According to statistics, supplements help a third of all men who use them. Another effect of the natural composition of dietary supplements is the improvement of vascular tone. This also has a positive effect on potency. The indicated action is performed by drugs from the following list:
- Tribulus;
- Parity;
- Critical PCT;
- testoporject;
- Erectogenon;
- Prostatinol;
Testosterone in a pharmacy
The pharmacy sells different forms of this sex hormone. Each of them has its own features of use and advantages. The main types of testosterone preparations are:
- Capsules. They are the most comfortable form of all. Capsules are easier to digest by the body. The disadvantage is that the excretion is too fast, so the agent cannot maintain a normal glucose level for a long time.
- Ointments and gels. Compared to capsules and tablets, this form is more effective. The hormone from the ointment or gel penetrates the blood faster. The disadvantage is that with prolonged use, allergic reactions are possible.
- plasters. They are glued to any part of the body, more often specifically to the scrotum. The active ingredient in contact with the skin quickly penetrates into the blood. The downside is the possibility of rashes.
- Injections. Thanks to injections, the steroid enters the body bypassing the digestive system, which is why the active component of the drug enters the bloodstream faster.
- Implants. They are small capsules placed in the abdomen. They are applied after being embedded under the skin. The normal level of the sex hormone is maintained for 6 months.
Nebido
Medicine made in Germany. It is an oily solution for injection. The active ingredient in the composition is testosterone undecanoate. The amount in one ampoule is 4 ml. The indication for use is the need to raise the level of the sex hormone of the same name. Other features of using Nebido:
- Dosage. Makes 1 ampoule of the drug, i.e. 1 g daily. The injection is administered immediately after opening. Do it as slowly as possible.
- duration of treatment. Equals 3-4 months, taking into account the patient's condition.
- Contraindications. Include androgen-dependent malignant tumor of the breast or prostate carcinoma, hypercalcemia, hypersensitivity to the composition, female sex, liver tumor.
- Side effects. Manifested by all body systems. more common reaction in the form of acne and pain at the place of possession.
Androgel
French testosterone preparation, produced in the form of a gel. The active substance in it is the hormone of the same name. Each sachet of disposable gel contains 25 or 50 mg of the active ingredient. Auxiliary substances are carbopol, sodium hydroxide, ethanol, water. The tool has a pronounced androgenic and anabolic effect. It has the only indication for use - replacement therapy for hypogonadism in case of testosterone deficiency. Before using the medicine, you need to study its main features:
- How to use. The gel is used externally at the same time every day. The dosage is 5 g. It can be adjusted by a doctor, but not more than 10 g. The gel is applied to clean and dry skin of the shoulders or abdomen, after which it is left to dry for 3-5 minutes. It is not recommended to use the product on the genitals.
- Course of androgen therapy. Determined by the doctor.
- Contraindications. They are hypersensitivity to the composition, heart failure, tumors, prostate cancer, epilepsy, arterial hypertension.
- Side effects. Possible acne, irritation and erythema at the site of use, increased pressure, paresthesia, dizziness, diarrhea, alopecia.
Testosterone Propionate
Judging by the reviews of doctors and patients, this tool is one of the best. It is a solution of an oily liquid with a specific odor. An auxiliary component in it is ethyl oleate. Testosterone is sold in 1 ml ampoules. The drug has an anabolic and androgenic effect. As a result of this influence, the development and functions of the external genital organs and secondary male sexual characteristics are stimulated. Other features of this testosterone preparation:
- Indications for use. Includes prostate dystrophy, impotence, acromegaly, sexual underdevelopment, androgen deficiency, oligospermia, mastopathy, uterine myoma, endometriosis.
- Dosage and duration of treatment. Determined according to the disease. in most cases, the patient is prescribed 1 ml for intramuscular injection.
- Contraindications. You can not use the drug for prostate hyperplasia, myocardial infarction, gynecomastia, diabetes, prostate cancer.
- Side effects. Increased sexual arousal, atrophy of the mammary glands, pastosity of the face, masculinization in women are possible.
Sustanon
Sustanon 250 contains several types of testosterone - cypionate, enanthate, propionate. Additionally, it contains peanut butter, benzyl alcohol and nitrogen. The solution is available in colorless glass ampoules. The drug is used in replacement therapy in case of primary and secondary hypogonadism. The solution is injected deep intramuscularly, 1 ml every 3 weeks. Side effects when using high doses: prostate cancer, neoplasms, fluid retention, polycythemia. Sustanon 250 contraindications are:
- age less than 3 years;
- suspected prostate or breast cancer;
- sensitivity to the components of the drug.
Andriol
Testosterone preparations are often available in tablet form. For example, the drug Andriol. These tablets and capsules are well tolerated by patients and do not suppress testosterone production. The medicine makes up for his lack. Indications for use are:
- hypopituitarism;
- postcastration syndrome;
- infertility;
- endocrine impotence;
- menopausal symptoms in men;
- masculinization in transsexuals.
The dosage of the drug is 120-160 mg. Reception is carried out within 2-3 weeks. as side effects, there may be a closure of bone growth zones, premature puberty, an increase in the frequency of erections. Contraindications to taking Andriol are:
- lactation;
- pregnancy;
- intolerance to components;
- carcinoma of the prostate or breast.
Omnadren
The basis of the drug Omnadren 250 is a mixture of testosterone esters. The release form is an oily solution for injection. Indications for use are:
- impotence;
- infertility;
- postkartsionny syndrome;
- eunuchoidism;
- oligospermia;
- hypopituitarism;
- male menopause;
- lack of androgens.
The average dosage is 1 ml of the product. The drug is injected 1 time in 28 days deep into the gluteal muscle. Side effects may occur in relation to the endocrine, reproductive, digestive, circulatory and nervous systems. contraindications to the use of Omnadren:
- hypercaluria;
- suspected carcinoma of the prostate or breast;
- pregnancy and lactation;
- renal, hepatic or heart failure.
Parity
In the category of dietary supplements for increasing testosterone, Parity can be distinguished. It is based on the extract of Eurycoma longifolia roots, Yohimbe bark, Maral antlers, Ginger rhizome and nicotinamide. The composition contains vitamin E, magnesium stearate. The principle of action is to stimulate the body to produce its own sex hormone. Use this effect in case of complaints about:
- erectile dysfunction;
- decreased libido;
- lack of vitamin E, zinc and Nicotinamide.
Adults are prescribed 1 capsule daily with food. The course of therapy lasts 15 days. After application, allergic reactions are possible. A contraindication to taking Paritet is only individual intolerance to the components. Cases of drug overdose were not observed. It is only possible to increase the listed side effects.
Tribulus
The basis of this remedy is the plant Tribulus Terrestris. Through chemical reactions, a food extract is obtained from raw materials, which is classified as a highly effective preparation. Take the drug 1-3 times every day after meals. The maximum allowable daily dose is 1250 mg. Indications for use are:
- male infertility;
- diseases of the genitourinary system;
- to increase libido;
- menopause;
- impotence.
When treated with Tribulus, acne, digestive disorders and blood pressure jumps may occur. You can not take the drug when:
- diseases of the cardiovascular system;
- prostate hypertrophy;
- renal failure;
- individual intolerance to the components of the drug.
Vitrix
Another powerful testosterone booster is Vitrix. The tool belongs to the category of sports nutrition. The Tribulus plant also acts as the basis, but the drug itself is produced using a different technology. Formulated with a special liquid blend of phyto-nutrients including Eurycoma longifolia, Blackberry, Common Oat and Epidmedium. Take the drug should be 3 capsules in the morning and evening. Vitrix is contraindicated in:
- pregnancy;
- lactation;
- individual intolerance to the components;
- under 18 years of age.
The price of testosterone preparations
The cost of medicines and dietary supplements is determined by the type of product, its manufacturer and place of purchase. You can buy testosterone tablets for men in Moscow and St. Petersburg at the following prices.
Testosterone is a male hormone. If it is not enough, it must be replenished. For example, testosterone tablets can be used. If there is not enough testosterone in the body, then many male functions will be weakened or suspended. There are alternative ways to replenish testosterone (injections, for example). But before taking these pills or injecting, you should understand what testosterone is and how it affects the body.
male sex hormone
As already mentioned, testosterone is a male sex hormone. But one should not think that women do not have such a hormone. It's just that its amount in a woman's body is much less. Testosterone is involved in the formation and strengthening of bone tissue, protein synthesis and has an anabolic effect. That is why the body of a man, as a rule, is characterized by a more powerful skeleton, developed muscles and muscle mass and less perception of pain. These properties of testosterone formed the basis of many hormonal drugs, which are prescribed for women in case of corresponding diseases.
For some diseases, testosterone tablets or testosterone-based hormonal preparations can be prescribed not only for men, but also for women. This is due to the fact that some diseases arise precisely because of the weakness of the skeleton or a violation of the process of protein synthesis, where testosterone is indispensable.
Testosterone is produced from cholesterol by cells of the adrenal cortex, in small amounts by the ovaries in women, and by cells of the testes in men. And if women need this hormone in minimal amounts (in the absence of corresponding diseases), then for men it is a vital hormone. In addition to the synthesis of proteins and the formation of bone tissue, it stimulates the functioning of the reproductive system.
Read also:
List of exercises for prostatitis.
natural and synthetic
Testosterone tablets can be divided into two large types: natural and synthetic. Natural testosterone is made from legumes. It differs from synthetic in that it is not very well absorbed by the body in tablet form. The fact is that testosterone is a hormone that partially breaks down when it enters the acidic environment of the stomach. To prevent this from happening, special protective additives are required. When injected, the degree of digestibility is much higher. But even here it should be noted that testosterone, which is produced by the body of each person, has individual characteristics. Therefore, even the injection method of administration does not guarantee complete digestibility in the body. Synthetic testosterone tablets in this regard are more effective than natural ones. It contains special substances that protect it in the acidic environment of the stomach before being absorbed into the blood.
Comparing the effects of synthetic and natural testosterone, you should know that natural, due to its low digestibility, does not create a stressful state for the body. It is absorbed scantily, and therefore gradually accustoms the body to increasing its dose in the blood. Synthetic can create a hormonal shock if used carelessly. Its dosage should be significantly less with a gradual increase to normal. Therefore, from the financial side, it may be more efficient to take synthetic, but in this case you need to be more careful with dosages.
Dosage
Take pills containing testosterone, should be strictly prescribed by the doctor and in the dosages that he indicated. If you replace one tablet with another, it is not enough to recalculate the hormone content in proportion, it is important to know what kind of testosterone it is - synthetic or natural. If you replace synthetic tablets with tablets with the same natural content and take them in the same mode, it is likely that the course of treatment will be extended by an insufficient amount of absorbed hormone. There is a chance to delay the treatment of the disease and "heal" the body (to create a period of adaptation to the drug for the disease, then at these doses the treatment will no longer be effective). And if, on the contrary, you replace natural testosterone with tablets with the same concentration of synthetic, then it may well be that the body will fail as a result of excess testosterone.
Excess testosterone leads to excessive irritability, mental excitability, even aggressiveness. On a chemical and biological level, this will result in the release of additional "calming" hormones into the blood, which can interfere with effective treatment, one of the elements of which was the introduction of testosterone.
Injections are much cheaper than the tablet form, because in this case, less dosage of testosterone is required due to better absorption. But the method of administering testosterone through injections requires a qualified nurse who knows how to make this kind of injection, sterile syringes and sufficient control of the situation on the part of doctors (the absorption of the drug is high, and there may be unforeseen situations related to the individual condition at the time of injection). If a person is away from the doctor (for example, in the country), then the tablet form looks much more preferable and safer.
Characteristic
Do not think that the introduction of testosterone into the body will make a person more courageous. Hormones should not be overestimated. If a man thinks he doesn't look or act masculine enough, it's not a testosterone problem. This is a psychological moment that must be addressed by psychological measures (going in for sports, developing a life line of behavior, etc.). Solving psychological problems by chemical methods is the last thing. It should be understood that the concept of "male hormones" is conditional, it characterizes not a psychotype, but only a physiological affiliation. And that is not absolutely, but only to a greater extent. Women also produce this hormone. But the main thing is that this hormone is not the only thing that distinguishes a man from a woman. There are many differences, not only in physiological terms, but also in the chemical composition of the blood, for example.
Purpose
Unreasonable self-administration of testosterone can lead to very bad consequences, for example, with the liver. The doctor, prescribing hormonal drugs, is guided not only by the task of defeating the disease, but also by the principle of "do no harm." You don't have to play with hormones. In our body, everything is very precisely verified, folded and adjusted. Each change entails a chain of changes throughout the body. Everything is interconnected. If you want to be more courageous, work on it. Something needs to be changed in the way of life, and not in the chemical composition of the blood.
The introduction of any drug leads to changes in the work of all (or many) organs. Qualitative changes happen slowly. Establishing work and treatment takes time and a competent approach.
In relation to bodybuilding, testosterone is one of the most important elements that help in building the body. It is often used, but only in injectable form. The low digestibility of tablet forms makes it impossible to use them for this sport. You can, of course, take handfuls of pills, but in this case there is a chance of worsening liver function. It should be understood that what did not enter the bloodstream in the form of testosterone will enter the body in a different form. But first it will be filtered by the liver. At the moment, such hormonal preparations have been developed that are absorbed into the blood before entering the liver. They are called prohormones. These drugs are good because they do not create swelling of the liver, are well absorbed and do not suppress the natural production of testosterone in the body.
Testosterone- a special drug, if not privileged. Synthetic, artificially obtained copy of the male sex hormone. The scheme of testosterone, its structure was unraveled back in 1935. Experiments on the hormone began to be carried out in the forties, and they continue to this day. Testosterone is a well-studied hormone with a pronounced anabolic effect, i.e. promotes the development and growth of muscle mass, burning fat and adding physical strength. Testosterone is available in various variations and dosages, there are injections of 50 mg, there are also huge doses of 250 mg, there is even tablet testosterone in dosages from 25 to 50 mg. Perhaps testosterone is so popular due to its study, everyone is well aware of its features and side effects, its effect on both the female body and the male body.
It would seem that testosterone is so studied and so simple, but it still remains the main headache for anti-doping companies. There is a problem of defining, identifying, testosterone in the blood of an athlete at competitions and this serious problem has not been solved to this day.
Testosterone constantly circulates through the blood channels, metabolizing and transforming into 17-keto metabolites, mainly into androsterone. It is these metabolites that are detected in the analysis of urine. The level of the drug in the urine is extremely small. Synthetic testosterone behaves exactly like natural testosterone, and therefore it is extremely difficult to distinguish it from artificial. It was also not possible to measure the peaks and falls of testosterone, so the drug remained an undetectable steroid until 1984.
Testosterone and its problems.
The first to take on the difficult task of identifying testosterone athletes was Manfred Donike, professor and founder of the Institute for Biochemistry of Sports in Cologne. He managed to synthesize the MSTFA reagent, which easily detected artificial testosterone and similar drugs (linked testosterone molecules into compounds that were easy to detect). Also, the professor was the first to guess not to measure the concentration of testosterone and its ratio to the concentration of epitestosterone (when using steroids, this ratio changed in the opposite direction). To announce his discovery, Donica needed thousands of analyzes to prove its truth. And he received such tests for artificial testosterone, somehow he managed to get unopened urine samples from the 1980 Olympics in Moscow. With the help of them, the professor managed to conduct detailed studies and already in 1984, at the Los Angeles Olympics, introduce his analysis for the content of artificial testosterone into widespread use.
There were also opponents, many did not want this analysis to appear in big-time sports. Their main argument was false negative results ( testosterone use for some reason did not always affect the change in the level of T / E, thus giving false test results). Basically, this defect was manifested in athletes with a congenital high content of E (mainly athletes from Asian countries).
Later it turned out that there are also false positive test results, the so-called false doping test, which athletes often had to deal with. Two such cases have been identified. Athletes from Norway and Australia had a stable unchangeable level of T / E, which constantly revealed their analyzes as positive. The athletes were observed for a long time, but their T/E levels did not change. Subsequently, it turned out that a large number of people, 1 in 2.5 thousand, have this feature (studies conducted in Sweden and Switzerland).
Doping test of testosterone athletes.
To confirm positive samples, some revolutionary method was needed, everyone understood this, even Donike himself. The professor made another attempt, he decided to measure the steroid profile, in this case, when taking testosterone, easily detectable distortions appeared. It was for the search for these distortions that Donike undertook. But, as in the case before, this test also had its drawbacks. Perhaps the most important of these was that doping test was relevant only for men, while in women it did not reveal any anomalies or deviations from the norm. And secondly, such distortions could appear under the influence of stressful situations, overtraining, or prolonged illness.
This method has not become a new revolution in the fight against testosterone. However, a couple of times, profile measurements nevertheless declared themselves. GDR sprint star Katrin Krabbe was caught in one of these tests. In 1992, at the Olympic Games in Barcelona, all of her tests were immediately positive. Catherine herself said that it was a fraud and fraud on the part of her ill-wishers. As it turned out in the end, it is almost impossible to prove her guilt. To put it simply, before she entered the study of her doping test, she traveled the world for several weeks and proved that no substitution was possible. But this is not the end, in the same year another urine sample was taken, doping tests, what was the surprise of the athlete when clenbuterol was found in her urine (in 1992, not yet a prohibited drug). The Olympic Committee decided to add clenbuterol to the list of prohibited drugs and sentence Crabbe to 4 years of deprivation of a sports license. From the ethical point of view, this is not the right decision, however, from the point of view of the law, it is possible and fair (by the way, Crabbe is not the only one who was caught using clenbuterol, in the same year, together with Crabbe, Grit Breuer, also an athlete from GDR).
The list of testosterone doping is huge and is expanding every year, even now many athletes do not hesitate to use it. Perhaps the most famous sports star on this list is Ben Johnson. In 1993, he received a life ban. His urinalysis for doping testosterone showed an increased ratio of T to E (the ratio at the time of sampling was at the level of 9, while his, i.e. natural, was on the border of three).
Artificial testosterone and athletes affected by it.
Another star on this list is Dennis Mitchell, a US runner (Olympic and world champion, former world record holder in the 100m sprint). In 1998, his urinalysis showed an unprecedented level of testosterone. However, in his case, everything worked out, the athlete was acquitted, but I want to note that after this incident, Mitchell's career came to naught, his results worsened every year and, in the end, he had to leave the bigger sport.
Also worth remembering is Mary Dekker-Slaney, a famous long-distance runner. The list of her achievements is huge, which is only worth the victory over Soviet athletes in 1983. In 1996, the athlete was caught using testosterone. As a result, the athlete missed the selection for the Olympics and, as a result, the Olympics itself, even despite the protection from NIKE and many athletes from the United States. By the way, along with Mary, Sandra Farmer-Patrick (a 400-meter hurdler) also got caught on testosterone. I forgot to say, both athletes received lengthy disqualifications.
There are also Soviet athletes on this list. At least two. These are Ukrainian Alexander Bagach (heavyweight, shot putter) and Russian Irina Belova (athletics, heptathlon). Alexander Bagach caused the USSR national team to miss the World Cup (taking 2nd place in the selection, after Bagach's disqualification they rolled back to third), and Irina was completely disqualified for the maximum possible period for her misconduct, i.e. for 4 years.
As you can easily see from the above examples, testosterone does not spare anyone, athletes of different sexes and different orientations, from runners to weightlifters, fall under its influence. Perhaps the reason for this is the effectiveness of synthetic testosterone, because all the athletes who took it inconspicuously achieved results in sports. However, there is one “BUT” here, the long-term use of artificial testosterone causes the so-called estrogen problem, well researched, but no less dangerous. Proved that artificial testosterone with its long-term use, it stops the production of natural testosterone and increases the synthesis of estrogens. This leads to the manifestation of female fat deposits, an increase in the timbre of the voice, etc., it comes to the point that a man's chest begins to grow. Ask bodybuilders, anyone will tell you that this is the problem. But here, too, a solution has been found, today on the market you will not find any antiestrogens and estrogen inhibitors. Now science really does not sleep.
Synthetic testosterone and its natural analogue.
Finally, I want to talk about the lawsuits and the athletes accused of using testosterone. Now most of the steroid drugs and supplements are able to cause an increase in the ratio of T to E. There have been such cases that athletes have been condemned for using steroid supplements, even though they are quietly sold in pharmacies, like regular vitamins or aspirin. But after all, if you think about it, the athlete did not take either the artificial version or testosterone, he took the drug, which is freely available. Multiple trials have already bothered the Americans so much that they generally removed synthetic testosterone from the list of prohibited drugs in sports such as Basketball and Rugby.
The same problem with nandrolone, doping tests that determine synthetic testosterone, give a positive result, and the athlete claims that he did not take nandrolone, he just ate a couple of pills, vitamins bought at a pharmacy. In this case, Dieter Baumann and Merlin Otti immediately come to mind. As a result, Merlin Otti was acquitted, a long trial decided that, despite the high content of nandrolone and increased testosterone, the athlete could be released, because the concentration of urine was also high, and if the concentration of urine was reduced, then the content of nandrolone would drop to the permitted results.
What can I add here, but actually nothing. I am only sure that during the life of Manfred Donike, such controversial situations would not have arisen. However, time flies and sports along with it. I put an end to this, although no, in Sydney in the year 2000, a new method was used to detect testosterone, multiple studies have shown its effectiveness. Let's hope that this is not the end, because we all love clean sports.
In conclusion, it is important to say that testosterone-based preparations, including the steroid testosterone propionate, you can easily purchase from our store. Only high-quality pharmacology at reasonable prices!
Source: AthleticPharma.com
And women play an important role in organisms. This male hormone is necessary for the formation of bones, protein synthesis, and under its influence, the full functioning of the genital organs occurs.
Sometimes, when an underestimated level of this hormone in the body is detected, doctors prescribe the use of testosterone tablets.
How are tablets classified?
Testosterone tablets are divided into synthetic and natural.
Testosterone of natural origin
The hormone of natural origin is produced on the basis of plant components:
What is this hormone responsible for?
- soy;
- legumes.
In laboratories, a number of hormones are created that are similar in composition to the substance that is produced in the male body. This type of testosterone is produced in micron doses and may not be fully absorbed in the body. Testosterone (micronized) has a long exposure period, which makes it possible to maintain the level of the male hormone for 24 hours.
At the same time, increased sexual desire appears, the body is filled with energy, patients improve their general health, tone, and bone tissue gains density. It is worth noting that taking testosterone (micronized) is manifested by side effects in the form of increased pressure, water retention in the body, and an increase in the amount of harmful testosterone in plasma.
Synthetic Testosterone
Types of tablet hormone
Testosterone (synthetic) is different from the natural substance. The first difference is the chemical composition, due to which it is quickly absorbed in the body through the bloodstream. After using a testosterone tablet, a pronounced effect is noted. When taking synthetic testosterone in tablet form, significant jumps of the hormone in human plasma occur. With a sharp increase in hormone levels after use, patients may experience a feeling of anxiety, aggression, irritability, muscle spasms, and headaches. When the hormonal level decreases in men, weakness is felt.
Among the huge number of pills for increasing testosterone, there is a list of the most frequently recommended drugs by specialists.
Methyltestosterone
Testosterone tablets. Means of synthetic origin, does not have complete decay and is completely absorbed in the body. Among the side effects noted violation of the liver, this is one of the reasons why the drug is not in wide demand in medicine.
Andrakson
Effective remedyThis type of hormone is called prohormones. The active substances of the drug do not disturb the water balance in the body (they do not retain fluid), and most importantly, Androxon does not suppress the natural production of testosterone by the body. Athletes taking this drug confirm that the drug does not have a significant anabolic effect. In men involved in sports, who took advantage of this testosterone, there was an increase in muscle mass, with an increase in its volume. The growth of muscle tissue is observed only after the use of 240 mg of the daily dosage of the drug. However, this dose may cause side effects.
- impaired spermatogenesis;
- male infertility;
- eunuchoidism;
- with impotence.
Synthetic testosterone is also allowed to be taken by the female sex:
- during menopausal disorders;
- with myomas;
- osteoporosis.
The drug is prescribed only by a specialist who individually selects the dosage according to the age category, the patient's condition and gender differences. The use of the product is allowed without deviations from the instructions. The daily dose is 120-160 mg. Therapeutic therapy is prescribed for a three-week period, then the treatment regimen passes into maintenance therapy (daily dose of 120 mg).
Before the profile specialist prescribes the use of this remedy, the patient's prostate gland is examined. During the treatment course, control of hormonal levels and hematocrit (the number of red blood cells) is required.
Possible side effects
When synthetic testosterone is prescribed as hormone therapy to replace a deficiency of this substance, side effects are possible in patients:
Side effects
- anisocytosis;
- erythrocytosis;
- increased libido;
- frequent erections;
- reduced volume of ejaculate.
With prolonged use of Andrakson, a decrease in the production of seminal fluid appears, tumors may appear in the prostate, water retention by the body.
Some men have manifestations of alopecia areata, gynecomastia, dizziness, manifestations of nausea, and progressive sleep apnea.
Who is contraindicated in replacement therapy
Contraindications for the use of synthetic testosterone include cancer patients who have tumors in the prostate gland. Do not take the drug to men with hyperplasia, erythrocytosis, heart failure, severe course, kidney pathology.
The female sex is forbidden to take drugs while carrying a child, breastfeeding, with oncological processes of the mammary gland.
Andriol
Active substanceAnother name for the drug may be undecanoate. The tool is available in tablets, it does not have such a negative effect on the liver. This is due to the absorption of the drug by the intestines and the transition to the lymph.
The drug does not increase estrogen, so there is no risk of fluid accumulation in the body. The drug has no negative impact on the natural production of testosterone. The tool is known as an effective medical care for infertility, impaired spermatogenesis, eunuchoidism, impotence associated with hormonal imbalance, reduced libido, chronic menopause, oligospermia.
Women are prescribed a remedy for:
- disturbed climacteric course;
- osteoporosis;
- uterine fibroids;
- endometriosis;
- menopause;
- hyperestrogenism;
- malignant tumors in the mammary glands.
Mestirolone
Analogues of this drug are Proviron, Wistinon. These drugs do not have destructive properties for the liver, do not subject to aromatization, which explains the use of the drug for obesity with increased estrogen activity.
Natural remedies that increase the production of natural testosterone by the body itself
Food supplement
- Tribestan - the drug has a positive effect on the synthesis in the body. The product contains extracts of Tribulus. The tool is used to stabilize the production of natural testosterone, as a stabilizer of the urinary and reproductive systems in the female and male body. The drug is prescribed in the treatment of infertility, to stimulate endocrine processes, strengthen bone tissue, and regulate calcium metabolism.
- Testogenon is available in capsule form. In its composition it has an extract of the bark of pygeum, ginseng rhizomes, yohimba, a vitamin and mineral complex. The drug is recommended to be taken to increase potency with the stabilization of health in the reproductive system. The drug is often used in recovery from infectious and inflammatory diseases, and also as a prophylactic for people who live or work in a harmful environment.
- Tribulus - This product contains tribulus extract. The plant does a good job of normalizing the production of hormones by the pituitary gland, and also restores hormonal balance, in general.
Athletes very often use herbal remedies to gain muscle volume.
From year to year, any organism physiologically wears out. Biological processes slow down, internal organs lose their functionality, hormone synthesis decreases, and the body begins to fail. This is especially reflected in the male body, in which a deficiency of the male hormone can lead to androgen deficiency.
Therefore, doctors recommend treatment in the form of hormone replacement therapy. As a rule, intramuscular injections of testosterone cypionate are one of the types of effective drugs for men. Preparations containing testosterone are sold in any pharmacy - in the public domain and without a prescription.
Testosterone preparations on the pharmacological market are presented as:
- testosterone injections;
- Testosterone tablets - oral route of administration;
- Testosterone patch and testosterone gel - transdermal method of application;
- Suspension of testosterone;
- subcutaneous implants.
Artificial testosterone has not only a positive effect on the body of men, but also side effects from taking it. The most popular type of testosterone is the hormone in ampoules, namely testosterone cypionate. Hormone injections are divided into short, medium and long-acting injections according to their duration and effectiveness.
A short-acting testosterone, such as propionate, should be taken every 3 days. The hormonal course in this case will take a long period of time and will affect the unpleasant pain at the injection site.
Testosterone cypionate, as well as enanthate, sustanol and testosterone depot, are medium-acting drugs. They need to be pricked only once every 2-3 weeks. This is quite convenient, besides, the effectiveness of such drugs is greater than that of analogues.
Taking a long-acting hormone, such as nebido undeconate, has a fairly long interval - about 14 weeks. Throughout this time, the hormonal background in men is maintained in the normal range. This drug has virtually no side effects. The hormone, as a rule, is excreted from the blood without sharp fluctuations in the general hormonal background in the blood. This leads to the fact that men retain sexual function, libido and mood during this time. A significant disadvantage of undeconate is the price of the drug.
Popular hormone ester
Testosterone cypionate is the most affordable and popular activator of anabolic processes in the body of men today. Male hormone injections are presented in the form of an oil solution. A solo cycle of testosterone cypionate is combined with other anabolic drugs for weight gain.
The action of testosterone cypionate in the body is aimed at regulating physical and emotional processes. Thanks to this hormone, a voice and primary sexual characteristics are formed in men, muscle growth is activated, and sexual function is regulated. Solo course of the drug is indicated for use in sports pharmacology. The hormone activates the synthesis of nitrogen in the body, and this, in turn, is a natural process of growth and development of muscle protein.
The negative side of testosterone cypionate is that the esters of the drug are aromatized into estrogens. This negatively affects the body of men, since an excess of the female hormone leads to the formation of the mammary glands according to the female type, stagnation of fluid in the body, and excessive weight gain. Long-term use of testosterone cypionate leads to testicular atrophy in men and a decrease in libido.
Side effects can be prevented if the course of the drug is combined with excipients, namely Nolvadex and Clomid. It is also worth noting that after taking testosterone cypionate, there may be such negative consequences as increased secretion of sebum, dermatological diseases, and baldness. Side effects can be eliminated with the help of the drug propecia.
The course of testosterone cypionate is quite long. Injections of the drug should be done every week in the amount of 200-250 mg. To avoid side effects, you should not raise this dose to 800 mg.
To block the synthesis of the male hormone into estrogen, tamoxifen is additionally injected at a dosage of 10 mg per day or more, depending on how you feel. If the testosterone cycle lasts more than 4-5 weeks, then gonadotropin is additionally used.
The testosterone stimulator has a relatively low cost, which makes it affordable for all categories of the population.
Testosterone for oral administration
Testosterone tablets are intended for oral administration. Synthetic hormone is easily absorbed by the body. The course of the hormone in tablets helps to increase energy, the formation of sexual arousal in men, increases the density of bone and muscle mass, and also improves the physiological state of the body as a whole.
It is much easier and more convenient to use the male hormone in tablets. But, if testosterone injections are rapidly absorbed in the gastrointestinal tract, then the half-life of the tablet preparation is much longer.
The pharmacological market presents the male hormone in tablets in the following range: methyltestosterone, androlala, testoral, andriol, androxon, virigen. Despite the convenience of using the drug in the form of tablets, they are still rarely recommended for use. This is due to the low effect of testosterone. The course of the drug in a high dosage does not entail a significant change in the physiological state of the body. For example, the increase in muscle mass in this case will be only 7%, while testosterone injections form muscles by 40%.
For men with androgen deficiency solo, a course of testosterone tablets is not recommended for use. The only possible form of treatment is a combination of oral hormone and the steroid nandrolone.
Water solution
Testosterone injections are indicated for use in the form of an aqueous solution of the hormone. Testosterone suspension has a number of side effects. Basically, testosterone suspension is used in sports pharmacology in men involved in heavy sports. The advantage of suspensions is that their complete disintegration and utilization from the body occur within a day. While other synthetic analogues of the hormone do not have such an effect.
Testosterone suspension is one of the very first artificially derived anabolic steroids. Since the molecular structure of the drug is presented without ether in the composition, the testosterone suspension in 100 mg is presented exclusively in the form of a pure substance without impurities. Hormone analogs cannot demonstrate the same performance, since the same enanthate from 100% of the substance gives the body only 73%, everything else disappears with the ether.
Instructions for use of the drug testosterone suspension:
- The minimum half-life of the active substance;
- Accelerated anabolic effect on the body, manifested in the first 24 hours from the moment of injection;
- High androgenic activity of the drug.
Testosterone suspension has a number of side effects that are not hidden by any instructions for use. The drug is prone to cause dermatological diseases, gynecomastia, increased sebum secretion. Also, an aqueous solution of testosterone has a negative effect on the liver. To avoid adverse reactions of the body, it is necessary to inject each dose of the drug in a new place. To reduce pain, the hormone in suspension is combined with vitamin B12.
Analogues of the artificial male hormone are also presented in the form of a gel and a patch containing a small amount of the hormone. They are prescribed to patients diagnosed with hypogonadism (low testosterone levels). An increase in the level of the hormone occurs while the gel penetrates the epithelium.
Testosterone patches are recommended for the elderly to prevent androgen deficiency.
A significant disadvantage of transdermal testosterone preparations is their short-term effect - only 24 hours. Then you need to glue a new patch or apply the gel to the skin. Gel Androgel and plaster Androderm have a high cost, which makes them inaccessible to the general population. Taking hormonal drugs should be carried out only after a doctor's prescription. Self-medication can lead to adverse effects.